Gregorio Valencia Parera-rekin lankidetzan egindako argitalpenak (9)

2020

  1. Calorimetric Studies of Binary and Ternary Molecular Interactions between Transthyretin, Aβ Peptides, and Small-Molecule Chaperones toward an Alternative Strategy for Alzheimer's Disease Drug Discovery

    Journal of Medicinal Chemistry, Vol. 63, Núm. 6, pp. 3205-3214

2019

  1. Radiochemical examination of transthyretin (TTR) brain penetration assisted by iododiflunisal, a TTR tetramer stabilizer and a new candidate drug for AD

    Scientific Reports, Vol. 9, Núm. 1

2017

  1. Insights on the Interaction between Transthyretin and Aβ in Solution. A Saturation Transfer Difference (STD) NMR Analysis of the Role of Iododiflunisal

    Journal of Medicinal Chemistry, Vol. 60, Núm. 13, pp. 5749-5758

  2. Role of the sugar moiety on the opioid receptor binding and conformation of a series of enkephalin neoglycopeptides

    Bioorganic and Medicinal Chemistry, Vol. 25, Núm. 7, pp. 2260-2265

2015

  1. Influence of polar side chains modifications on the dual enkephalinase inhibitory activity and conformation of human opiorphin, a pain perception related peptide

    Bioorganic and Medicinal Chemistry Letters, Vol. 25, Núm. 22, pp. 5190-5193

  2. Modulation of the Interaction between a Peptide Ligand and a G Protein-Coupled Receptor by Halogen Atoms

    ACS Medicinal Chemistry Letters, Vol. 6, Núm. 8, pp. 872-876

2012

  1. Structure-activity relationship study of opiorphin, a human dual ectopeptidase inhibitor with antinociceptive properties

    Journal of Medicinal Chemistry, Vol. 55, Núm. 3, pp. 1181-1188

2011

  1. Synthesis, biological evaluation and structural characterization of novel glycopeptide analogues of nociceptin N/OFQ

    Organic and Biomolecular Chemistry, Vol. 9, Núm. 17, pp. 6133-6142

2009

  1. Synthesis, conformation, and biological characterization of a sugar derivative of morphine that is a potent, long-lasting, and nontolerant antinociceptive

    Journal of Medicinal Chemistry, Vol. 52, Núm. 9, pp. 2656-2666