Farmacia y Ciencias de los Alimentos
Departamento
CONCEPCION ESTIBALIZ
ALONSO PEREZ
PROFESORADO TITULAR DE UNIVERSIDAD
Publicaciones en las que colabora con CONCEPCION ESTIBALIZ ALONSO PEREZ (13)
2022
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Multicomponent Synthesis of Unsaturated γ-Lactam Derivatives. Applications as Antiproliferative Agents through the Bioisosterism Approach: Carbonyl vs. Phosphoryl Group
Pharmaceuticals, Vol. 15, Núm. 5
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Synthesis of hybrid phosphorated indenoquinolines and biological evaluation as topoisomerase I inhibitors and antiproliferative agents
Bioorganic and Medicinal Chemistry Letters, Vol. 57
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The design and discovery of topoisomerase I inhibitors as anticancer therapies
Expert Opinion on Drug Discovery, Vol. 17, Núm. 6, pp. 581-601
2021
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A patent review of topoisomerase I inhibitors (2016–present)
Expert Opinion on Therapeutic Patents, Vol. 31, Núm. 6, pp. 473-508
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Design, synthesis and cytotoxic evaluation of diphenyl(quinolin-8-yl)phosphine oxides
Tetrahedron Letters, Vol. 70
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Hybrid quinolinyl phosphonates as heterocyclic carboxylate isosteres: Synthesis and biological evaluation against topoisomerase 1b (top1b)
Pharmaceuticals, Vol. 14, Núm. 8
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Simple and fast dna based sensor system for screening of small-molecule compounds targeting eukaryotic topoisomerase 1
Pharmaceutics, Vol. 13, Núm. 8
2020
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Fused 1,5-Naphthyridines: Synthetic Tools and Applications
Molecules (Basel, Switzerland), Vol. 25, Núm. 15
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Synthesis of novel hybrid quinolino[4,3-b][1,5]naphthyridines and quinolino[4,3-b][1,5]naphthyridin-6(5H)-one derivatives and biological evaluation as topoisomerase I inhibitors and antiproliferatives
European Journal of Medicinal Chemistry, Vol. 195
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Synthetic strategies, reactivity and applications of 1,5-naphthyridines
Molecules, Vol. 25, Núm. 14
2019
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Antileishmanial activity of new hybrid tetrahydroquinoline and quinoline derivatives with phosphorus substituents
European Journal of Medicinal Chemistry, Vol. 162, pp. 18-31
2018
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Novel topoisomerase I inhibitors. Syntheses and biological evaluation of phosphorus substituted quinoline derivates with antiproliferative activity
European Journal of Medicinal Chemistry, Vol. 149, pp. 225-237
2014
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Synthesis and biological evaluation of 1,5-naphthyridines as topoisomerase I inhibitors. A new family of antiproliferative agents
Current Topics in Medicinal Chemistry, Vol. 14, Núm. 23, pp. 2722-2728