Química Orgánica I
Departamento
Aarhus University
Århus, DinamarcaPublicaciones en colaboración con investigadoras/es de Aarhus University (22)
2023
-
Gel-Free Tools for Quick and Simple Screening of Anti-Topoisomerase 1 Compounds
Pharmaceuticals, Vol. 16, Núm. 5
2022
-
Synthesis of hybrid phosphorated indenoquinolines and biological evaluation as topoisomerase I inhibitors and antiproliferative agents
Bioorganic and Medicinal Chemistry Letters, Vol. 57
2021
-
A dual-sensor-based screening system for in vitro selection of tdp1 inhibitors
Sensors, Vol. 21, Núm. 14
-
Fused chromeno and quinolino[1,8]naphthyridines: Synthesis and biological evaluation as topoisomerase I inhibitors and antiproliferative agents
Bioorganic and Medicinal Chemistry, Vol. 40
-
Hybrid quinolinyl phosphonates as heterocyclic carboxylate isosteres: Synthesis and biological evaluation against topoisomerase 1b (top1b)
Pharmaceuticals, Vol. 14, Núm. 8
-
Simple and fast dna based sensor system for screening of small-molecule compounds targeting eukaryotic topoisomerase 1
Pharmaceutics, Vol. 13, Núm. 8
2020
-
Novel phosphine sulphide gold(i) complexes: topoisomerase I inhibitors and antiproliferative agents
Dalton Transactions, Vol. 49, Núm. 23, pp. 7852-7861
-
Synthesis of novel hybrid quinolino[4,3-b][1,5]naphthyridines and quinolino[4,3-b][1,5]naphthyridin-6(5H)-one derivatives and biological evaluation as topoisomerase I inhibitors and antiproliferatives
European Journal of Medicinal Chemistry, Vol. 195
2019
-
Straightforward synthesis and biological evaluation as topoisomerase I inhibitors and antiproliferative agents of hybrid Chromeno[4,3-b][1,5]Naphthyridines and Chromeno[4,3-b][1,5]Naphthyridin-6-ones
European Journal of Medicinal Chemistry, Vol. 178, pp. 752-766
2018
-
Novel topoisomerase I inhibitors. Syntheses and biological evaluation of phosphorus substituted quinoline derivates with antiproliferative activity
European Journal of Medicinal Chemistry, Vol. 149, pp. 225-237
2017
-
Advantages of an optical nanosensor system for the mechanistic analysis of a novel topoisomerase i targeting drug: A case study
Nanoscale, Vol. 9, Núm. 5, pp. 1886-1895
2016
-
Reply to comment on "radicalicity: A scale to compare reactivities of radicals"
Chemical Physics Letters
-
Synthesis and biological evaluation of indeno[1,5]naphthyridines as topoisomerase i (TopI) inhibitors with antiproliferative activity
European Journal of Medicinal Chemistry, Vol. 115, pp. 179-190
2015
-
Radicalicity: A scale to compare reactivities of radicals
Chemical Physics Letters, Vol. 618, pp. 99-101
2007
-
Bisoxazoline-Lewis acid-catalyzed direct-electron demand oxo-hetero-Diels-Alder reactions of N-oxy-pyridine aldehyde and ketone derivatives
Journal of Organic Chemistry, Vol. 72, Núm. 1, pp. 240-245
-
Treatment of vibronic interactions using variational methods for nuclear motion
AIP Conference Proceedings
-
Variational calculation of static and dynamic vibrational nonlinear optical properties
Journal of Chemical Physics, Vol. 127, Núm. 8
2006
-
A simple asymmetric organocatalytic approach to optically active cyclohexenones
Chemical Communications, pp. 4928-4930
-
Bis(oxazoline) lewis acid catalyzed aldol reactions of pyridine N-oxide aldehydes-synthesis of optically active 2-(1-hydroxyalkyl)pyridine derivatives: Development, scope, and total synthesis of an indolizine alkaloid
Chemistry - A European Journal, Vol. 12, Núm. 13, pp. 3472-3483
-
One-pot organocatalytic domino Michael-aldol and intramolecular S N2 reactions. Asymmetric synthesis of highly functionalized epoxycyclohexanone derivatives
Journal of the American Chemical Society, Vol. 128, Núm. 16, pp. 5475-5479