Publications by the researcher in collaboration with H. Konno (22)

2022

  1. New pharmaceuticals approved by FDA in 2020: Small-molecule drugs derived from amino acids and related compounds

    Chirality, Vol. 34, Núm. 1, pp. 86-103

2021

  1. Asymmetric Synthesis of N-Fmoc-(S)-7-aza-tryptophan via Alkylation of Chiral Nucleophilic Glycine Equivalent

    European Journal of Organic Chemistry, Vol. 2021, Núm. 21, pp. 2962-2965

  2. Asymmetric Synthesis of α-Difluorinated β-Amino Sulfones through Detrifluoroacetylative Mannich Reactions

    European Journal of Organic Chemistry, Vol. 2021, Núm. 21, pp. 3035-3038

  3. Asymmetric synthesis of (S)-3-methyleneglutamic acid and its N-Fmoc derivative via Michael addition–elimination reaction of chiral glycine Ni (II) complex with enol tosylates

    Chirality, Vol. 33, Núm. 3, pp. 115-123

  4. Asymmetric synthesis of the two enantiomers of β-phosphorus-containing α-amino acids: Via hydrophosphinylation and hydrophosphonylation of chiral Ni(ii)-complexes

    Organic Chemistry Frontiers, Vol. 8, Núm. 10, pp. 2190-2195

  5. Comparative study of different chiral ligands for dynamic kinetic resolution of amino acids

    Chirality, Vol. 33, Núm. 10, pp. 685-702

  6. Peptidomimetics and peptide-based blockbuster drugs

    Current Organic Chemistry, Vol. 25, Núm. 14, pp. 1627-1658

  7. Tailor-Made Amino Acids in Pharmaceutical Industry: Synthetic Approaches to Aza-Tryptophan Derivatives

    Chemistry - A European Journal, Vol. 27, Núm. 70, pp. 17510-17528

  8. Tailor-made amino acids in the design of small-molecule blockbuster drugs

    European Journal of Medicinal Chemistry, Vol. 220

2020

  1. Asymmetric Mannich reactions of (S)-N-tert-butylsulfinyl-3,3,3-trifluoroacetaldimines with yne nucleophiles

    Beilstein Journal of Organic Chemistry, Vol. 16, pp. 2671-2678

  2. Asymmetric Synthesis of 4,4-(Difluoro)glutamic Acid via Chiral Ni(II)-Complexes of Dehydroalanine Schiff Bases. Effect of the Chiral Ligands Structure on the Stereochemical Outcome

    ChemistryOpen, Vol. 9, Núm. 1, pp. 93-96

  3. Asymmetric Synthesis of Tailor-Made Amino Acids Using Chiral Ni(II) Complexes of Schiff Bases. An Update of the Recent Literature

    Molecules (Basel, Switzerland), Vol. 25, Núm. 12

  4. Asymmetric synthesis of (S)-α-(octyl)glycine via alkylation of Ni(II) complex of chiral glycine Schiff base

    Chirality, Vol. 32, Núm. 12, pp. 1354-1360

  5. Kitamura electrophilic fluorination using HF as a source of fluorine

    Molecules, Vol. 25, Núm. 9

  6. Large-Scale Synthesis of the Glycine Schiff Base Ni(II) Complex Derived from (S)- A nd (R)-N-(2-Benzoyl-4-chlorophenyl)-1-[(3,4-dichlorophenyl)methyl]-2-pyrrolidinecarboxamide

    Organic Process Research and Development, Vol. 24, Núm. 2, pp. 294-300

  7. Michael addition reactions of chiral glycine Schiff base Ni (II)-complex with 1-(1-phenylsulfonyl)benzene

    Chirality, Vol. 32, Núm. 6, pp. 885-893

  8. Synthesis of Ahod Moiety of Ralstonin A Using Amino Acid Schiff Base Ni(II)-Complex Chemistry

    Helvetica Chimica Acta, Vol. 103, Núm. 7

  9. Tailor-made amino acid-derived pharmaceuticals approved by the FDA in 2019

    Amino Acids, Vol. 52, Núm. 9, pp. 1227-1261

2019

  1. Asymmetric synthesis of (2S,3S)-3-Me-glutamine and (R)-allo-threonine derivatives proper for solid-phase peptide coupling

    Amino Acids, Vol. 51, Núm. 3, pp. 419-432

  2. Convenient synthesis of racemic 4,4-difluoro glutamic acid derivatives via Michael-type additions of Ni(II)-complex of dehydroalanine Schiff bases

    Journal of Fluorine Chemistry, Vol. 227