Publicaciones (21) Publicaciones de ENDIKA MARTIN ENCINAS

2024

  1. Antileishmanial Effect of 1,5- and 1,8-Substituted Fused Naphthyridines

    Molecules, Vol. 29, Núm. 1

  2. Aza-Povarov Reaction. A Method for the Synthesis of Fused Tetracyclic Chromeno[4,3-d]pyrido[1,2-a]pyrimidines

    Journal of Organic Chemistry, Vol. 89, Núm. 2, pp. 1099-1107

  3. Synthesis, biological and computational evaluation of novel cyanomethyl vinyl ether derivatives

    Frontiers in Pharmacology, Vol. 15

2023

  1. Kanptotezina eta haren deribatuak minbiziaren aurkako borrokan: Topoisomerasa I inhibitzaileak

    Ekaia: Euskal Herriko Unibertsitateko zientzi eta teknologi aldizkaria, Núm. 44, pp. 127-136

2022

  1. Hydrogen sulphide-triggered theranostic prodrugs based on the dynamic chemistry of tetrazines

    Chemical Communications, Vol. 58, Núm. 36, pp. 5518-5521

  2. The design and discovery of topoisomerase I inhibitors as anticancer therapies

    Expert Opinion on Drug Discovery, Vol. 17, Núm. 6, pp. 581-601

2021

  1. A dual-sensor-based screening system for in vitro selection of tdp1 inhibitors

    Sensors, Vol. 21, Núm. 14

  2. A patent review of topoisomerase I inhibitors (2016–present)

    Expert Opinion on Therapeutic Patents, Vol. 31, Núm. 6, pp. 473-508

  3. Dynamic Nucleophilic Aromatic Substitution of Tetrazines

    Angewandte Chemie - International Edition, Vol. 60, Núm. 34, pp. 18783-18791

  4. Fused chromeno and quinolino[1,8]naphthyridines: Synthesis and biological evaluation as topoisomerase I inhibitors and antiproliferative agents

    Bioorganic and Medicinal Chemistry, Vol. 40

  5. Naphthyridine derivatives induce programmed cell death in naegleria fowleri

    Pharmaceuticals, Vol. 14, Núm. 10

  6. Tetrazine Dynamic Covalent Polymer Networks

    Macromolecules, Vol. 54, Núm. 22, pp. 10428-10434

2020

  1. Fused 1,5-Naphthyridines: Synthetic Tools and Applications

    Molecules (Basel, Switzerland), Vol. 25, Núm. 15

  2. Novel phosphine sulphide gold(i) complexes: topoisomerase I inhibitors and antiproliferative agents

    Dalton Transactions, Vol. 49, Núm. 23, pp. 7852-7861

  3. Synthesis of novel hybrid quinolino[4,3-b][1,5]naphthyridines and quinolino[4,3-b][1,5]naphthyridin-6(5H)-one derivatives and biological evaluation as topoisomerase I inhibitors and antiproliferatives

    European Journal of Medicinal Chemistry, Vol. 195

  4. Synthetic strategies, reactivity and applications of 1,5-naphthyridines

    Molecules, Vol. 25, Núm. 14

2019

  1. Antileishmanial activity of new hybrid tetrahydroquinoline and quinoline derivatives with phosphorus substituents

    European Journal of Medicinal Chemistry, Vol. 162, pp. 18-31

  2. Straightforward synthesis and biological evaluation as topoisomerase I inhibitors and antiproliferative agents of hybrid Chromeno[4,3-b][1,5]Naphthyridines and Chromeno[4,3-b][1,5]Naphthyridin-6-ones

    European Journal of Medicinal Chemistry, Vol. 178, pp. 752-766

2018

  1. Novel topoisomerase I inhibitors. Syntheses and biological evaluation of phosphorus substituted quinoline derivates with antiproliferative activity

    European Journal of Medicinal Chemistry, Vol. 149, pp. 225-237

  2. Synthesis of novel antiproliferative hybrid bis-(3-indolyl)methane phosphonate derivatives

    European Journal of Medicinal Chemistry, Vol. 158, pp. 874-883