LUIS FELIPE
CALLADO HERNANDO
PROFESORADO PLENO
Trinity College Dublin
Dublín, IrlandaPublicaciones en colaboración con investigadoras/es de Trinity College Dublin (12)
2021
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Di-aryl guanidinium derivatives: Towards improved α2-Adrenergic affinity and antagonist activity
European Journal of Medicinal Chemistry, Vol. 209
2017
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Thiophene/thiazole-benzene replacement on guanidine derivatives targeting α2-Adrenoceptors
European Journal of Medicinal Chemistry, Vol. 138, pp. 38-50
2016
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Substituted conformationally restricted guanidine derivatives: Probing the α2-adrenoceptors’ binding pocket
European Journal of Medicinal Chemistry, Vol. 123, pp. 48-57
2015
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α2-adrenoceptor antagonists: Synthesis, pharmacological evaluation, and molecular modeling investigation of pyridinoguanidine, pyridino-2-aminoimidazoline and their derivatives
Journal of Medicinal Chemistry, Vol. 58, Núm. 2, pp. 963-977
2014
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Guanidine-based α2-adrenoceptor ligands: Towards selective antagonist activity
European Journal of Medicinal Chemistry, Vol. 82, pp. 242-254
2013
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Antidepressant-like properties of three new α2-adrenoceptor antagonists
Neuropharmacology, Vol. 65, pp. 13-19
2008
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Guanidine and 2-aminoimidazoline aromatic derivatives as α2-adrenoceptor antagonists. 2. Exploring alkyl linkers for new antidepressants
Journal of Medicinal Chemistry, Vol. 51, Núm. 11, pp. 3304-3312
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Novel synthesis and pharmacological evaluation as α2-adrenoceptor ligands of O-phenylisouronium salts
Bioorganic and Medicinal Chemistry, Vol. 16, Núm. 17, pp. 8210-8217
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PHARMACOLOGICAL EVALUATION OF GUANIDINE AND 2-AMINOIMIDAZOLINE AROMATIC DERIVATIVES AS alpha(2)-ADRENOCEPTOR ANTAGONISTS
METHODS AND FINDINGS IN EXPERIMENTAL AND CLINICAL PHARMACOLOGY
2007
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Guanidine and 2-aminoimidazoline aromatic derivatives as α2-adrenoceptor antagonists, 1: Toward new antidepressants with heteroatomic linkers
Journal of Medicinal Chemistry, Vol. 50, Núm. 18, pp. 4516-4527
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On the search of new I2-IBS aliphatic ligands: Bis-guanidino carbonyl derivatives
Bioorganic and Medicinal Chemistry Letters, Vol. 17, Núm. 21, pp. 6009-6012
2002
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I2-imidazoline binding site affinity of a structurally different type of ligands
Bioorganic and Medicinal Chemistry, Vol. 10, Núm. 5, pp. 1525-1533