FRANCISCO JAVIER
PALACIOS GAMBRA
PROFESORADO EMERITO
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Aarhus University
Århus, DinamarcaPublicaciones en colaboración con investigadoras/es de Aarhus University (10)
2021
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A dual-sensor-based screening system for in vitro selection of tdp1 inhibitors
Sensors, Vol. 21, Núm. 14
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Fused chromeno and quinolino[1,8]naphthyridines: Synthesis and biological evaluation as topoisomerase I inhibitors and antiproliferative agents
Bioorganic and Medicinal Chemistry, Vol. 40
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Hybrid quinolinyl phosphonates as heterocyclic carboxylate isosteres: Synthesis and biological evaluation against topoisomerase 1b (top1b)
Pharmaceuticals, Vol. 14, Núm. 8
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Simple and fast dna based sensor system for screening of small-molecule compounds targeting eukaryotic topoisomerase 1
Pharmaceutics, Vol. 13, Núm. 8
2020
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Novel phosphine sulphide gold(i) complexes: topoisomerase I inhibitors and antiproliferative agents
Dalton Transactions, Vol. 49, Núm. 23, pp. 7852-7861
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Synthesis of novel hybrid quinolino[4,3-b][1,5]naphthyridines and quinolino[4,3-b][1,5]naphthyridin-6(5H)-one derivatives and biological evaluation as topoisomerase I inhibitors and antiproliferatives
European Journal of Medicinal Chemistry, Vol. 195
2019
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Straightforward synthesis and biological evaluation as topoisomerase I inhibitors and antiproliferative agents of hybrid Chromeno[4,3-b][1,5]Naphthyridines and Chromeno[4,3-b][1,5]Naphthyridin-6-ones
European Journal of Medicinal Chemistry, Vol. 178, pp. 752-766
2018
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Novel topoisomerase I inhibitors. Syntheses and biological evaluation of phosphorus substituted quinoline derivates with antiproliferative activity
European Journal of Medicinal Chemistry, Vol. 149, pp. 225-237
2017
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Advantages of an optical nanosensor system for the mechanistic analysis of a novel topoisomerase i targeting drug: A case study
Nanoscale, Vol. 9, Núm. 5, pp. 1886-1895
2016
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Synthesis and biological evaluation of indeno[1,5]naphthyridines as topoisomerase i (TopI) inhibitors with antiproliferative activity
European Journal of Medicinal Chemistry, Vol. 115, pp. 179-190