Publications (72) Publications de CONCEPCION ESTIBALIZ ALONSO PEREZ

2024

  1. Antileishmanial Effect of 1,5- and 1,8-Substituted Fused Naphthyridines

    Molecules, Vol. 29, Núm. 1

  2. Aza-Povarov Reaction. A Method for the Synthesis of Fused Tetracyclic Chromeno[4,3-d]pyrido[1,2-a]pyrimidines

    Journal of Organic Chemistry, Vol. 89, Núm. 2, pp. 1099-1107

  3. Synthesis, biological and computational evaluation of novel cyanomethyl vinyl ether derivatives

    Frontiers in Pharmacology, Vol. 15

2023

  1. Efficient AntiMycolata Agents by Increasing the Lipophilicity of Known Antibiotics through Multicomponent Reactions

    Antibiotics, Vol. 12, Núm. 1

  2. Gel-Free Tools for Quick and Simple Screening of Anti-Topoisomerase 1 Compounds

    Pharmaceuticals, Vol. 16, Núm. 5

  3. The Intramolecular Povarov Tool in the Construction of Fused Nitrogen-Containing Heterocycles

    Topics in Current Chemistry, Vol. 381, Núm. 4

2022

  1. Hydrogen sulphide-triggered theranostic prodrugs based on the dynamic chemistry of tetrazines

    Chemical Communications, Vol. 58, Núm. 36, pp. 5518-5521

  2. Multicomponent Synthesis of Unsaturated γ-Lactam Derivatives. Applications as Antiproliferative Agents through the Bioisosterism Approach: Carbonyl vs. Phosphoryl Group

    Pharmaceuticals, Vol. 15, Núm. 5

  3. Synthesis of hybrid phosphorated indenoquinolines and biological evaluation as topoisomerase I inhibitors and antiproliferative agents

    Bioorganic and Medicinal Chemistry Letters, Vol. 57

  4. The design and discovery of topoisomerase I inhibitors as anticancer therapies

    Expert Opinion on Drug Discovery, Vol. 17, Núm. 6, pp. 581-601

2021

  1. A dual-sensor-based screening system for in vitro selection of tdp1 inhibitors

    Sensors, Vol. 21, Núm. 14

  2. A patent review of topoisomerase I inhibitors (2016–present)

    Expert Opinion on Therapeutic Patents, Vol. 31, Núm. 6, pp. 473-508

  3. Design, synthesis and cytotoxic evaluation of diphenyl(quinolin-8-yl)phosphine oxides

    Tetrahedron Letters, Vol. 70

  4. Fused chromeno and quinolino[1,8]naphthyridines: Synthesis and biological evaluation as topoisomerase I inhibitors and antiproliferative agents

    Bioorganic and Medicinal Chemistry, Vol. 40

  5. Hybrid quinolinyl phosphonates as heterocyclic carboxylate isosteres: Synthesis and biological evaluation against topoisomerase 1b (top1b)

    Pharmaceuticals, Vol. 14, Núm. 8

  6. Naphthyridine derivatives induce programmed cell death in naegleria fowleri

    Pharmaceuticals, Vol. 14, Núm. 10

  7. Simple and fast dna based sensor system for screening of small-molecule compounds targeting eukaryotic topoisomerase 1

    Pharmaceutics, Vol. 13, Núm. 8

2020

  1. Fused 1,5-Naphthyridines: Synthetic Tools and Applications

    Molecules (Basel, Switzerland), Vol. 25, Núm. 15

  2. New Challenges in Drug Discovery – July 8–11, 2019, Vitoria-Gasteiz, Spain

    ChemMedChem

  3. Novel phosphine sulphide gold(i) complexes: topoisomerase I inhibitors and antiproliferative agents

    Dalton Transactions, Vol. 49, Núm. 23, pp. 7852-7861