Publications (73) Publications de JESUS MANUEL DE LOS SANTOS RUIZ

2024

  1. Diastereoselective ZnCl2-Mediated Joullié–Ugi Three-Component Reaction for the Preparation of Phosphorylated N-Acylaziridines from 2H-Azirines

    Molecules, Vol. 29, Núm. 5

  2. Exploring the Reactivity of Rigid 1-Azadienes Derived from Methylene γ-Lactams. Applications to the Stereoselective Synthesis of Spiro-γ-Lactams

    Journal of Organic Chemistry, Vol. 89, Núm. 13, pp. 9502-9515

2023

  1. Chiral self-recognition in a bispericyclic cyclodimerisation reaction of 1-azadienes

    Organic Chemistry Frontiers, Vol. 10, Núm. 24, pp. 6103-6111

  2. Synthesis and Characterization of a New Series of Bis(allylic-α-aminophosphonates) under Mild Reaction Conditions

    Molecules, Vol. 28, Núm. 12

  3. Synthesis of Fused Nitrogenated Heterocycles: Intramolecular Povarov Reaction

    Advances in Organic Synthesis (Bentham Science Publishers), pp. 40-111

  4. The Intramolecular Povarov Tool in the Construction of Fused Nitrogen-Containing Heterocycles

    Topics in Current Chemistry, Vol. 381, Núm. 4

2022

  1. Multicomponent Synthesis of Unsaturated γ-Lactam Derivatives. Applications as Antiproliferative Agents through the Bioisosterism Approach: Carbonyl vs. Phosphoryl Group

    Pharmaceuticals, Vol. 15, Núm. 5

  2. Sc(OTf)3-Mediated [4 + 2] Annulations of N-Carbonyl Aryldiazenes with Cyclopentadiene to Construct Cinnoline Derivatives: Azo-Povarov Reaction

    Journal of Organic Chemistry, Vol. 87, Núm. 17, pp. 11583-11592

2021

  1. Phosphinotripeptidic inhibitors of leucylaminopeptidases

    International Journal of Molecular Sciences, Vol. 22, Núm. 10

  2. Synthesis and antiproliferative activity of phosphorus substituted 4-cyanooxazolines, 2-aminocyanooxazolines, 2-iminocyanooxazolidines and 2-aminocyanothiazolines by rearrangement of cyanoaziridines

    Molecules, Vol. 26, Núm. 14

2020

  1. Copper-catalyzed synthesis of aziridines

    Copper in N-Heterocyclic Chemistry (Elsevier), pp. 1-48

  2. First synthesis of merged hybrids phosphorylated azirino[2,1-b]benzo[e][1,3]oxazine derivatives as anticancer agents

    European Journal of Medicinal Chemistry, Vol. 185

  3. New Challenges in Drug Discovery – July 8–11, 2019, Vitoria-Gasteiz, Spain

    ChemMedChem

  4. Synthesis of α-Aminophosphonic Acid Derivatives Through the Addition of O- and S-Nucleophiles to 2H-Azirines and Their Antiproliferative Effect on A549 Human Lung Adenocarcinoma Cells

    Molecules (Basel, Switzerland), Vol. 25, Núm. 15

2019

  1. Multicomponent reactions (MCRs): A useful access to the synthesis of benzo-fused γ-lactams

    Beilstein Journal of Organic Chemistry, Vol. 15, pp. 1065-1085

  2. Natural deep eutectic solvents in the hetero-Diels–Alder approach to bis(indolyl)methanes

    Monatshefte fur Chemie, Vol. 150, Núm. 7, pp. 1275-1288

  3. Reaction of phosphinyl nitrosoalkenes with electron-rich heterocycles

    Phosphorus, Sulfur and Silicon and the Related Elements, Vol. 194, Núm. 4-6, pp. 545-549

  4. Synthesis and biological evaluation of cyanoaziridine phosphine oxides and phosphonates with antiproliferative activity

    European Journal of Medicinal Chemistry, Vol. 163, pp. 736-746

2018

  1. Catalytic Asymmetric Darzens and Aza-Darzens Reactions for the Synthesis of Chiral Epoxides and Aziridines

    ChemCatChem, Vol. 10, Núm. 22, pp. 5092-5114

  2. Multicomponent reactions in the synthesis of γ-Lactams

    Synthesis (Germany), Vol. 50, Núm. 23, pp. 4539-4554